Alpha-blockers

Adrainolitics wani rukuni ne na sunadaran da ke shafar wasu masu karɓar adrenergic. Dangane da abin da waɗannan abubuwa ke shafar adrenoreceptors, an raba su zuwa beta da alpha-blockers. Shirye-shiryen da aka tsara akan su an tsara shi ne a kan yaki da nau'o'in kwayoyin zuciya, tsarin daji, idan akwai yanayin ƙwayar cuta kuma don daidaita yanayin.

Shiryawa Alpha-blockers

Akwai manyan magunguna guda biyu.

Masu jefa kuri'a marasa zaɓi

Abubuwa da ke damuwa da ayyukan adenoreceptors postynaptic, wanda ya haifar da fadada lumen daga cikin jirgi da kuma saukowa daga matsin lamba, da kuma yaduwancin norepinephrine.

Babban wakili na rukuni na farko shine Fentolamine, wanda tasirinsa shine kara yawan tasoshin ruwa. Lokacin da aka gudanar da abu a cikin intravenously, ana samun sakamako a cikin minti goma sha biyar.

A magani, an yi amfani da magani yanzu da wuya, amma ana iya tsara shi don:

Wasu wakilan wannan rukuni:

Zaɓin Alpha-1-adrenoblockers

Wadannan abubuwa sune mafi girman aiki da tsawon lokaci. Suna da sakamako masu tasiri akan matakin cholesterol cikin jini, saboda haka rage hadarin bunkasa atherosclerosis. Bugu da ƙari, abubuwa ba su shafi tasirin sukari ba, kar ka ƙara matsa lamba kuma bambanta a cikin ƙananan ƙwayoyin cutar.

Zaɓin alpha-blockers zaɓaɓɓen sun hada da jerin jerin kwayoyi:

Ta hanyar tasirin su, wadannan kwayoyi sun fi gaban Fentolamine. Muhimmin tasirin su shine rage rage ta hanyar rage maye gurbin ƙarancin jini. Abubuwan da suka fara fara bayyana bayan kimanin sa'a daya bayan rikici.

Shaida don amfani da Alpha-adrenoblockers

Ka yi la'akari da ilimin warkewar wasu ƙwayoyi:

  1. Tare da cututtukan kwayoyin halitta na jini (cutar Raynaud), a cikin maganin warkar da raunuka da kuma decubitus, kuma a cikin kula da pheochromocytomas, Fentolamine da Tropafen an tsara su.
  2. Matakan farko na ci gaban adenoma prostate suna bi da su tare da Prozazin, wanda ya inganta fitowar fitsari.
  3. Alfa-1-adrenoblockers sun kasance mafi yawan su a hauhawar jini. Suna fadada tasoshin (daga mafi ƙanƙanci zuwa mafi girma), don haka rage matsa lamba. Ragewa daga matsa lamba yana haifar da wani mahimmanci a cikin kaya a kan myocardium, wanda ke sa wadannan kwayoyi suyi tasiri a cikin infarction m .
  4. Don maganin lokaci mai tsawo, ana amfani da Prazonin da Doxazine.
  5. Dukkanin abubuwan da aka ba da kyauta suna da Fentolamin da Prazonin.
  6. Ana amfani da diabergergotamine don ƙaura, da magungunan ƙwayar cuta da ƙwayar cuta.

Contraindications Alpha-blockers

Kada ku bada magunguna ga mutanen da suke da wadannan karkatarwa:

Abinda ya saba wa juna shi ne ciki.

Ana nuna alamun da ba'a so a matsayin: